Signaling peptide receptor
Signaling peptide receptor is a type of receptor which binds one or more signaling peptides or signaling proteins.
An example is the tropomyosin receptor kinase B (TrkB), which is bound and activated by the neurotrophic protein brain-derived neurotrophic factor (BDNF). Another example is the μ-opioid receptor (MOR), which is bound and activated by the opioid peptide hormone β-endorphin.
Adiponectin receptor
AdipoR1
- Agonists
- Peptide
- Adiponectin
 - ADP-355
 - ADP-399
 
 - Non-peptide
- AdipoRon
 - (–)-Arctigenin
 - Arctiin
 - Gramine
 - Matairesinol
 
 
 - Peptide
 - Antagonists
- Peptide
- ADP-400
 
 
 - Peptide
 
AdipoR2
- Agonists
- Peptide
- Adiponectin
 - ADP-355
 - ADP-399
 
 - Non-peptide
- AdipoRon
 - Deoxyschizandrin
 - Parthenolide
 - Syringing
 - Taxifoliol
 
 
 - Peptide
 - Antagonists
- Peptide
- ADP-400
 
 
 - Peptide
 
Angiotensin receptor
Bradykinin receptor
- Agonists
 - Antagonists
- FR-173657
 - Icatibant
 - LF22-0542
 
 
Calcitonin gene-related peptide receptor
- Agonists
 - Antagonists
- Atogepant
 - BI 44370 TA
 - CGRP (8-37)
 - MK-3207
 - Olcegepant
 - Rimegepant
 - SB-268262
 - Telcagepant
 - Ubrogepant
 
 - Antibodies
 
Cholecystokinin receptor
CCKA
- Agonists
 - Antagonists
- Amiglumide
 - Asperlicin
 - Devazepide
 - Dexloxiglumide
 - Lintitript
 - Lorglumide
 - Loxiglumide
 - Pranazepide
 - Proglumide
 - Tarazepide
 - Tomoglumide
 
 
CCKB
- Agonists
- Cholecystokinin
 - CCK-4
 - Gastrin
 - Pentagastrin (CCK-5)
 
 - Antagonists
- Ceclazepide
 - CI-988 (PD-134308)
 - Itriglumide
 - L-365,360
 - Netazepide
 - Proglumide
 - Spiroglumide
 
 
Unsorted
- Antagonists
- Nastorazepide
 
 
Corticotropin-releasing hormone receptor
CRF1
- Agonists
- Cortagine
 - Corticorelin
 - Corticotropin-releasing hormone
 - Sauvagine
 - Stressin I
 - Urocortin
 
 - Antagonists
- Antalarmin
 - Astressin-B
 - CP-154,526
 - Emicerfont
 - Hypericin
 - LWH-234
 - NBI-27914
 - NBI-74788
 - Pexacerfont
 - R-121919
 - TS-041
 - Verucerfont
 
 
CRF2
- Agonists
- Corticorelin
 - Corticotropin-releasing hormone
 - Sauvagine
 - Urocortin
 
 - Antagonists
- Astressin-B
 
 
Cytokine receptor
Endothelin receptor
- Agonists
- Endothelin 1
 - Endothelin 2
 - Endothelin 3
 - IRL-1620
 - Sarafotoxin
 
 - Antagonists
- A-192621
 - Ambrisentan
 - Aprocitentan
 - Atrasentan
 - Avosentan
 - Bosentan
 - BQ-123
 - BQ-788
 - Clazosentan
 - Darusentan
 - Edonentan
 - Enrasentan
 - Fandosentan
 - Feloprentan
 - Macitentan
 - Nebentan
 - Sitaxentan
 - Sparsentan
 - Tezosentan
 - Zibotentan
 
 
Galanin receptor
GAL1
GAL2
GAL3
- Agonists
 - Antagonists
- C7
 - Galantide (M15)
 - GalR3ant
 - HT-2157
 - M32
 - M35
 - M40
 - SNAP-37889
 - SNAP-398299
 
 
Growth hormone secretagogue receptor
Growth hormone receptor
Growth-hormone-releasing hormone receptor
Glucagon-like peptide receptor
GLP-1
- Agonists
- Albiglutide
 - Beinaglutide
 - Dulaglutide
 - Efpeglenatide
 - Exenatide
 - GLP-1
 - Langlenatide
 - Liraglutide
 - Lixisenatide
 - Oxyntomodulin
 - Pegapamodutide
 - Semaglutide
 - Taspoglutide
 
 
GLP-2
- Agonists
- Apraglutide
 - Elsiglutide
 - Glepaglutide
 - GLP-2
 - Teduglutide
 
 
Others
- Propeptides
 
Glucagon receptor
- Agonists
- Dasiglucagon
 - Glucagon
 - Oxyntomodulin
 
 - Antagonists
- Adomeglivant
 - L-168,049
 - LGD-6972
 
 - Propeptides
 
Gonadotropin-releasing hormone receptor
Gonadotropin receptor
Growth factor receptor
Insulin receptor
- Agonists
 - Antagonists
- BMS-754807
 - S661
 - S961
 
 - Kinase inhibitors
 - Antibodies
- Xentuzumab (against IGF-1 and IGF-2)
 
 
KiSS1-derived peptide receptor
- Agonists
- Kisspeptin (kisspeptin-54, metastin)
 - Kisspeptin-10
 - KISS1-305
 - MVT-602 (RVT-602, TAK-448)
 - TAK-683
 
 - Antagonists
- Kisspeptin-234
 
 
Leptin receptor
- Agonists
 
Melanin-concentrating hormone receptor
MCH1
- Agonists
- Melanin-concentrating hormone
 
 - Antagonists
- ATC-0065
 - ATC-0175
 - GW-803430
 - NGD-4715
 - SNAP-7941
 - SNAP-94847
 
 
MCH2
- Agonists
- Melanin-concentrating hormone
 
 
Melanocortin receptor
Neuropeptide FF receptor
- Agonists
- Neuropeptide AF
 - Neuropeptide FF
 - Neuropeptide SF (RFRP-1)
 - Neuropeptide VF (RFRP-3)
 
 - Antagonists
- BIBP-3226
 - RF9
 
 
Neuropeptide S receptor
Neuropeptide Y receptor
Y1
- Agonists
- Neuropeptide Y
 - Peptide YY
 
 - Antagonists
- BIBO-3304
 - BIBP-3226
 - BVD-10
 - GR-231118
 - PD-160170
 
 
Y2
- Agonists
- 2-Thiouridine 5'-triphosphate
 - Neuropeptide Y
 - Neuropeptide Y (13-36)
 - Peptide YY
 - Peptide YY (3-36)
 
 - Antagonists
- BIIE-0246
 - JNJ-5207787
 - SF-11
 
 
Y4
- Agonists
- GR-231118
 - Neuropeptide Y
 - Pancreatic polypeptide
 - Peptide YY
 
 - Antagonists
- UR-AK49
 
 
Y5
- Agonists
- BWX-46
 - Neuropeptide Y
 - Peptide YY
 
 - Antagonists
- CGP-71683
 - FMS-586
 - L-152,804
 - Lu AA-33810
 - MK-0557
 - NTNCB
 - Velneperit (S-2367)
 
 
Neurotensin receptor
NTS1
- Agonists
- Neurotensin
 - Neuromedin N
 
 - Antagonists
 
NTS2
- Agonists
- Neurotensin
 
 - Antagonists
 
Opioid receptor
Orexin receptor
Oxytocin receptor
Prolactin receptor
Parathyroid hormone receptor
- Agonists
 
Relaxin receptor
Somatostatin receptor
Tachykinin receptor
Thyrotropin-releasing hormone receptor
- Agonists
- Azetirelin
 - JTP-2942
 - Montirelin
 - Orotirelin
 - Posatirelin
 - Protirelin
 - Rovatirelin
 - RX-77368 (thymoliberin)
 - Taltirelin
 - TRH (TRF)
 
 
Thyrotropin receptor
- Agonists
 
Vasopressin receptor
Vasoactive intestinal peptide receptor and Pituitary adenylate cyclase-activating peptide
VIPR1
- Agonists
- Peptide
- Bay 55-9837
 - LBT-3393
 - PACAP
 - VIP
 
 
 - Peptide
 
VIPR2
- Agonists
- Peptide
- LBT-3627
 - PACAP
 - VIP
 
 
 - Peptide
 
PAC1
- Agonists
- PACAP
 - PACAP (1-27)
 - PACAP (1-38)
 
 - Antagonists
- PACAP (6-38)
 
 
Unsorted
- PHI
 - PHM
 - PHV
 
Others
- Endogenous
- Adrenomedullin
 - Apelin
 - Asprosin
 - Bombesin
 - Calcitonin
 - Carnosine
 - CART
 - CLIP
 - DSIP
 - Enteroglucagon
 - Formyl peptide
 - GALP
 - GIP
 - GRP
 - Integrin ligands
- collagens
 - fibrinogen
 - fibronectin
 - laminins
 - ICAM-1
 - ICAM-2
 - osteopontin
 - VCAM-1
 - vitronectin
 
 - Kininogens
 - Motilin
 - Natriuretic peptides 
- ANP
 - BNP
 - CNP
 - urodilatin
 
 - Nesfatin-1
 - Neuromedin B
 - Neuromedin N
 - Neuromedin S
 - Neuromedin U
 - Obestatin
 - Osteocalcin
 - Resistin
 - Secretin
 - Thymopoietin
 - Thymosins
 - Thymulin
 - Urotensin-II
 - VGF
 
 - Exogenous
- Lifitegrast (LFA-1 antagonist)
 
 
See also
References
External links
- Peptide+receptor at the U.S. National Library of Medicine Medical Subject Headings (MeSH)
 
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